| INHIBITOR | IN COMPLEXES | TYPE (ISOSTERE) | EC/RN NUMBER | REFERENCE |
| MVT101 | 4hvp |
|
12552-24-6 |
|
| A-74704 | 9hvp |
|
129467-45-4 |
|
| JG365 | 7hvp |
|
132748-20-0 |
|
| H261 | 2phv |
|
91464-97-0 |
|
| Acetylpepstatin | 1phv |
|
11076-29-2 |
|
| L-700,417 | 4phv |
|
|
|
| U-85548E | 8hvp |
|
124020-62-8 |
|
| SKF 108738 | 1hef,1siv |
|
144285-78-9 |
|
| SKF 107457 | 1heg |
|
144285-77-8 |
|
| U75875 | 1hiv |
|
112190-24-6 |
|
| SB204144 | 1hos |
|
141396-10-3 |
|
| GR123976 | 1hte |
|
|
|
| GR126045 | 1htf |
|
|
|
| BILA-398 | 2mip |
|
|
|
| EPNP | 2sam |
|
|
|
| U75875 | 1ivp |
|
|
|
| U92163 | 1ivq |
|
149607-21-6 |
|
| SB 206343 | 1hps |
|
|
|
| L-735,524 | 1hsg,1hsh |
|
|
|
| SB 203386 | 1sbg,1tcx,1tcw,
1bdl,1bdq,1bdr |
|
|
|
| A77003 | 1hvi,1hvs |
|
134878-17-4 |
|
| A78791 | 1hvj |
|
|
|
| A76928 | 1hvk,1hvc |
|
|
|
| A76889 | 1hvl |
|
134805-77-9 |
|
| GR137615 | 1htg |
|
|
|
| BILA -1906 | 1ida |
|
|
|
| BILA -2450 | 1idb |
|
||
| XK263 | 1hvr |
|
|
|
| SB203238 | 1hbv |
|
|
|
| CGP52820 | 1hii |
|
||
| VX-478 | 1hpv |
|
161814-49-9 |
|
| KNI-272 | 1hpx |
|
147318-81-8 |
|
| U095438 | 1upj |
|
||
| U100313 | 2upj |
|
|
|
| U096333 | 3upj,4upj |
|
||
| A79285 | 1dif |
|
||
| DMP323 | 1bve,1bvg,1mes,
1met,1meu |
|
151867-81-1 |
|
| U89360E | 1gnm,1gnn,1a9m |
|
162897-65-0 |
|
| Phe-Ile-Val | 1mtr |
|
||
| A98881 | 1pro |
|
|
|
| RO 31-8959 | 1hxb |
|
|
|
| BMS-182193 | 1odw,1odx |
|
|
|
| DMP450 | 1dmp,1mer |
|
|
|
| AHA006 | 1ajv |
|
||
| AHA001 | 1ajx |
|
||
| THK | 1aid |
|
||
| A84538 | 1hxw |
|
|
|
| BILA-N/A | 1jld |
|
||
| GLU-ASP-LEU | 1a30 |
|
||
| SDZ283-910 | 1a8g |
|
||
| SD146 | 1bv7,1bwb,hiv5dpm |
|
|
|
| XV638 | 1bv9,1bwa,hiv4dpm |
|
|
|
| RO 31-8558 | hiv2hlr |
|
||
| AG1001 | hiv1aug |
|
||
| AG1002 | hiv2aug |
|
||
| AG1004 | hiv3aug |
|
||
| LILLY765 | hiv1lll |
|
||
| I-BMS-01 | hiv1bms |
|
||
| I-BMS-02 | hiv2bms |
|
||
| BILA-2011 | hiv4bip |
|
||
| BILA-1780 | hiv5bip |
|
||
| Q8467 | hiv3dpm |
|