| SYSTEM |
|
|---|---|
| HIVdb File |
|
| PDB File |
|
| Company or Laboratory |
|
| Year |
|
| INHIBITOR (Type) |
|
| Composition of the Inhibitor (Substrate) or Summary Formula |
|
| Schematic Formula |
|
| Resolution |
|
| R factor |
|
| Space Group |
|
| Dimension of Elementary Cell |
|
| a,b,g
|
|
| Reference | H.L.Sham, C.Zhao, K.D.Stewart, D.A.Betterbenner, S.Lin, C.H.Park, X.P.Kong, W.Rosenbrook Junior, T.Herrin, D.Madigan, .D.J.Kempf, J.J.Platner, D.W.Norbeck; J.Med.Chem, 39, 392, 1996 |
| Comment | A picomolar inhibitor of HIV1 PR based on cyclic urea pioneered by DuPont Merck |