I)
Inhibitor (INH) - PR Complexes
A)OFFICIAL
RELEASES
| Inhibitor |
Type
of INH
|
Mutation(s)
|
PR
strain/isolate
|
PDB
file
|
HIV-db
file
|
|
|
amin-imide
peptide isostere
|
Q7K
|
SF strain
|
3aid
|
hiv8ucs
|
|
A77003
|
diol-isostere (R,S)
|
V82A
|
BH5 isolate
|
1hvs
|
hiv14nci
|
|
BMS-182193
|
|
A71T,V82A
|
HXB-2
isolate
|
1odx
|
hiv18nci
|
|
Cyclic
Phe-Ile?Val |
peptidomimetic
|
mutant
|
ARV2/SF2
isolate
|
1mtr
|
hiv2uba
|
|
DMP323
|
|
V82F,I84V
|
BH102
strain
|
1meu
|
hiv9dpm
|
|
DMP323
|
|
V82F
|
BH102 strain
|
1met
|
hiv8dpm
|
|
DMP323
|
|
I84V
|
BH102
strain
|
1mes
|
hiv7dpm
|
|
DMP323
|
cyclic
urea-type
|
C95A
|
HXB2
isolate
|
1bve
|
hiv1nid
|
|
DMP450
|
|
I84V
|
BH102
strain
|
1mer
|
hiv6dpm
|
|
SB203386
|
|
T31S,
L33V, E34T, E35G,M36I, S37E
|
|
1bdr
|
hiv12skb
|
|
SB203386
|
|
T31S, V32I, L33V, E34A,E35G, M36I, S37E, I47V, V82I
|
|
1bdq
|
hiv11skb
|
|
SB203386
|
|
T31S, V32I, L33V, E34A,E35G, M36I, S37E
|
|
1bdl
|
hiv10skb
|
|
SD146
|
|